SCHEMBL8138166

SCHEMBL8138166

NC(=O)Nc1ccc2ncccc2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
NPC1 O15118 4/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
HSD11B1 P28845 1/20 0.41
CYP3A4 P08684 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SYK P43405 1/20 0.41
RAB9A P51151 3/20 0.41
NR3C2 P08235 2/20 0.40
PABPC1 P11940 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4970115 0.85 KDM4E (0.46) KDM4EHSP90AA1HSP90AB1NPC1KMT2A
SCHEMBL27860315 0.83 CYP3A4 (0.47) KDM4EHSP90AA1HSP90AB1NPC1KMT2A
SCHEMBL15690239 0.83 KDM4E (0.66) KDM4EHSP90AA1HSP90AB1NPC1KMT2A
SCHEMBL8515227 0.79 KDM4E (0.70) KDM4EHSP90AA1HSP90AB1NPC1KMT2A
SCHEMBL31054265 0.78 KMT2A (0.68) NPC1KMT2AMEN1POLBMAPT
SCHEMBL2360527 0.77 NPC1 (0.65) NPC1KMT2AMAPTRAB9A
SCHEMBL7735807 0.77 KDM4E (0.51) KDM4ENPC1KMT2AMEN1POLB
Carbamic Acid SCHEMBL21437196 0.75 ALDH1A1 (0.50) KDM4ENPC1KMT2AMEN1POLB
SCHEMBL15223280 0.74 NCF1 (0.55) KDM4EHSP90AA1HSP90AB1NPC1POLB
SCHEMBL15726233 0.74 JAK2 (0.53) KDM4ENPC1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984967-A1 NAPHTHYRIDINE DERIVATIVES AND THEIR ANALOGUES INHIBITING CYTOMEGALOVIRUS BIOCHEM PHARMA INC (CA) 2000-03-15 EP disclosed
US-5945431-A VIRICIDE BIOCHEM THERAPEUTICS INCORPORATED (CA) 1999-08-31 US disclosed
WO-1997034894-A1 NAPHTHYRIDINE DERIVATIVES AND THEIR ANALOGUES INHIBITING CYTOMEGALOVIRUS BIOCHEM PHARMA INC. (CA) 1997-09-25 WO disclosed