SCHEMBL8139552

SCHEMBL8139552

CN(Cc1ccc(CNC(N)=O)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
TPSAB1 Q15661 4/20 0.45
GAA P10253 1/20 0.40
PRSS1 P07477 1/20 0.40
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
LSS P48449 1/20 0.39
EPHX2 P34913 2/20 0.39
NR1H4 Q96RI1 2/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
HTR2C P28335 1/20 0.38
SLC6A4 P31645 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3440346 0.83 KIF11 (0.43) CTSLCTSBCTSSGLS
SCHEMBL8526346 0.82 HTR2C (0.39) CTSLCTSBCTSSHDAC3HDAC1
SCHEMBL14829450 0.81 AOC3 (0.45) CTSLCTSBCTSSEPHX2NR1H4
SCHEMBL8139521 0.81 TPSAB1 (0.47) TPSAB1PRSS1CTSLCTSBCTSS
SCHEMBL2227505 0.81 HTR2C (0.41) CTSLCTSBCTSSEPHX2HDAC3
SCHEMBL23448763 0.81 HRH3 (0.44) CTSLCTSBCTSSLSSHDAC3
SCHEMBL23274094 0.80 HDAC3 (0.47) TPSAB1CTSLCTSBCTSSHDAC3
SCHEMBL30905374 0.79 L3MBTL1 (0.54) CYP2C9CYP2C19GAAEPHX2NR1H4
SCHEMBL2229917 0.79 MTOR (0.48) CTSLCTSBCTSSHDAC3HDAC1
SCHEMBL1935308 0.79 PPARG (0.46) CTSLCTSBCTSSHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114390-A AN ARGININAMIDE OR ORNITHINAMIDE COMPOUND AS TREATING MEMORY LOSS, MIGRAINE, SLEEP DISORDERS, PAIN, CARDIOVASCULAR DISEASES, SUBARACHNOIDAL BLEEDING, VASCULAR-HYPERTROPHIC CHANGES, CEREBRAL AND CORONARY VASOSPASMS KARL THOMAE GMBH (DE) 2000-09-05 US disclosed
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed