SCHEMBL8141015

SCHEMBL8141015

CN1CCc2c(-c3ccccc3S(=O)(=O)N(C)C)ccc(N)c2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
HTT P42858 1/20 0.39
HTR6 P50406 1/20 0.38
ALOX5AP P20292 5/20 0.38
FEN1 P39748 5/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
PDPK1 O15530 1/20 0.35
ROCK2 O75116 1/20 0.35
FES P07332 1/20 0.35
FER P16591 1/20 0.35
MARK3 P27448 1/20 0.35
FLT3 P36888 1/20 0.35
MAP4K2 Q12851 1/20 0.35
PKN2 Q16513 1/20 0.35
CDC42BPA Q5VT25 1/20 0.35
SLK Q9H2G2 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8126619 0.82 HTR6 (0.40) ALDH1A1HTTHTR6SMN1; SMN2HTR2A
SCHEMBL4394396 0.81 HTR6 (0.47) ALDH1A1HTTHTR6SMN1; SMN2HTR2A
SCHEMBL8133363 0.76 PDPK1 (0.40) ALDH1A1HTTHTR6SMN1; SMN2HTR2A
SCHEMBL14287257 0.73 PDPK1 (0.37) ALDH1A1HTTHTR6ALOX5APFEN1
Hydrochloric Acid SCHEMBL6613546 0.72 ALDH1A1 (0.42) ALDH1A1HTR2ACHRM2HTR1AADRA2A
SCHEMBL6608260 0.68 KDM4E (0.43) ALDH1A1HTR2ACHRM2HTR1AADRA2A
SCHEMBL8142621 0.68 CYP3A4 (0.43) ALDH1A1HTR1AKCNH2MAP4K1
SCHEMBL6611465 0.66 HDAC1 (0.38)
SCHEMBL13592435 0.66 GRIA1 (0.34) ALDH1A1CHRM2HTR1AADRA2ACHRM1
SCHEMBL8232020 0.65 CYP2C19 (0.39) ALDH1A1HTR2ACHRM2HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781285-B1 FUSED INDOLE AND QUINOXALINE DERIVATIVES, THEIR PREPARATION AND USE AS GLUTAMATE ANTAGONISTS NEUROSEARCH AS (DK) 2000-01-12 EP disclosed
US-5801174-A CEREBROVASCULAR DISORDERS NEUROSEARCH A/S (DK) 1998-09-01 US disclosed
WO-1996008495-A1 FUSED INDOLE AND QUINOXALINE DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1996-03-21 WO disclosed