SCHEMBL8232020

SCHEMBL8232020

Bc1ccc(N)c2c1CCN(C)C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
KDM4E B2RXH2 3/20 0.36
CYP2D6 P10635 3/20 0.36
CYP1A2 P05177 2/20 0.36
CHRNA7 P36544 1/20 0.36
ADRA1A P35348 4/20 0.36
ADRA2C P18825 3/20 0.36
ADRA2A P08913 3/20 0.36
ADRA2B P18089 2/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1B P35368 2/20 0.36
DRD1 P21728 2/20 0.34
DRD3 P35462 2/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD5 P21918 1/20 0.34
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3023510 0.80 ADRA2A (0.44) CYP2C19MAOAMAOBKDM4ECYP2D6
SCHEMBL17815212 0.78 CYP2C19 (0.39) CYP2C19MAOAMAOBKDM4ECYP2D6
SCHEMBL14402455 0.77 PNMT (0.43) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL4825313 0.77 SLC6A2 (0.42) CYP2C19MAOAMAOBKDM4ECYP2D6
SCHEMBL19705567 0.76 CYP2C19 (0.38) CYP2C19MAOAMAOBKDM4ECYP2D6
SCHEMBL8184550 0.76 CYP2C19 (0.38) CYP2C19MAOAMAOBKDM4ECYP2D6
SCHEMBL13875038 0.75 MAOA (0.44) MAOAMAOBKDM4ECYP2D6ADRA1A
SCHEMBL17197369 0.74 DRD1 (0.45) MAOAMAOBDRD1DRD3DRD2
Hydrochloric Acid SCHEMBL6613546 0.74 ALDH1A1 (0.42) MAOAMAOBKDM4ECYP2D6CYP1A2
SCHEMBL6608100 0.73 HRH4 (0.39) KCNH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007115408-A1 COMPOSITIONS AND METHODS FOR MODULATING GATED ION CHANNELS PAINCEPTOR PHARMA CORPORATION (CA) 2007-10-18 WO disclosed