SCHEMBL8141815

SCHEMBL8141815

Cc1ccc(S(=O)(=O)N(CCO)CC(O)Cc2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 3/20 0.47
MAPK1 P28482 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
MMP1 P03956 2/20 0.44
MMP2 P08253 2/20 0.44
MMP9 P14780 2/20 0.44
MMP8 P22894 2/20 0.44
MMP13 P45452 2/20 0.44
BACE1 P56817 2/20 0.43
CA12 O43570 2/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22750873 0.78 SMN1; SMN2 (0.62) CA9MAPK1ALDH1A1MAPTHTT
SCHEMBL9906199 0.74 MMP1 (0.45) CA9ALDH1A1MAPTBCHEACHE
SCHEMBL218536 0.73 SMN1; SMN2 (0.68) CA9MAPK1ALDH1A1MAPTMMP1
SCHEMBL16367398 0.73 ACHE (0.49) CA9ALDH1A1MAPTHTTBCHE
SCHEMBL9906204 0.73 MEN1 (0.52) CA9ALDH1A1MAPTHTTBCHE
SCHEMBL13558102 0.72 MMP1 (0.47) CA9ALDH1A1MAPTHTTBCHE
SCHEMBL15177296 0.72 SMN1; SMN2 (0.66) CA9MAPK1ALDH1A1MAPTMMP1
SCHEMBL8192690 0.72 SMN1; SMN2 (0.66) CA9MAPK1ALDH1A1MAPTMMP1
SCHEMBL6801648 0.71 MMP1 (0.61) ALDH1A1MMP1MMP2MMP9MMP8
SCHEMBL4401411 0.71 MAPT (0.58) CA9MAPK1ALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022966-A CONJUGATE COMPRISES A DOTA CHELATE COMPONENT, A BIOTIN COMPONENT AND A LINKER COMPONENT RESISTANT TO BIOTINIDASE CLEAVAGE NEORX CORPORATION (US) 2000-02-08 US disclosed
EP-0736035-A4 PRETARGETING METHODS AND COMPOUNDS NEORX CORP (US) 1999-09-01 EP disclosed
US-5847121-A Production of nitro-benzyl-dota via direct peptide cyclization NEORX CORPORATION (US) 1998-12-08 US disclosed
EP-0736035-A1 PRETARGETING METHODS AND COMPOUNDS NEORX CORPORATION (US) 1996-10-09 EP disclosed
US-5541287-A DIAGNOSIS USING CYCLIC TRIPEPTIDES WITH NITROBENZYL 1,4,7,10-TETRAAZACYCLODODECANE-N,N*,N**,N***TETRAACETIC ACID BIOTIN CONJUGATE FORMED BY ALKYLATION AND MULTISTAGE PROCESS NEORX CORPORATION (US) 1996-07-30 US disclosed
WO-1995015335-A2 PRETARGETING METHODS AND COMPOUNDS NEORX CORPORATION (US) 1995-06-08 WO disclosed