Treosulfan

Treosulfan

SCHEMBL8142

CS(=O)(=O)OCC(O)C(O)COS(C)(=O)=O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.43
ALDH1A1 P00352 2/20 0.43
TSHR P16473 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
MMP9 P14780 1/20 0.43
ALOX15 P16050 1/20 0.43
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Treosulfan SCHEMBL5399430 1.00 USP2 (0.43) USP2ALDH1A1TSHRKDM4ELMNA
Treosulfan SCHEMBL8466701 1.00 USP2 (0.43) USP2ALDH1A1TSHRKDM4ELMNA
SCHEMBL9359843 0.91 LMNA (0.37) USP2ALDH1A1TSHRKDM4ELMNA
SCHEMBL9359906 0.91 LMNA (0.37) USP2ALDH1A1TSHRKDM4ELMNA
SCHEMBL4951404 0.90 ALDH1A1 (0.40) USP2ALDH1A1TSHRKDM4ELMNA
Treosulfan SCHEMBL28276683 0.89 KDM4E (0.36) USP2ALDH1A1TSHRKDM4ELMNA
Treosulfan SCHEMBL28142583 0.89 KDM4E (0.36) USP2ALDH1A1TSHRKDM4ELMNA
Treosulfan SCHEMBL28086148 0.89 TSHR (0.65) USP2ALDH1A1TSHRKDM4ELMNA
SCHEMBL7621803 0.87 CA1 (0.39) USP2ALDH1A1TSHRKDM4ELMNA
SCHEMBL21815666 0.87 ALDH1A1 (0.39) USP2ALDH1A1TSHRKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 18018 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-20260102475-A1 REGIMEN FOR ENZYMATIC DESENSITISATION Hansa Biopharma AB (SE) 2026-04-16 US claimed
EP-3515892-B1 COMPOUNDS AND METHODS FOR IDO AND TDO MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC (US) 2026-04-15 EP claimed
US-20260091119-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF GLIOMA CELLIS AG (CH) 2026-04-02 US claimed
US-20260085061-A1 PHTHALAZINE DERIVATIVES AS PYRUVATE KINASE MODULATORS SITRYX THERAPEUTICS LIMITED (GB) 2026-03-26 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
EP-4257122-B1 LYOPHILISATE OF TREOSULFAN MEDAC GES FUER KLINISCHE SPEZIALPRAEPARATE MBH (DE) 2026-03-11 EP claimed
US-20260028400-A1 ANTI-ROR1 ANTIBODY AND USE THEREOF AIMED BIO INC (KR) 2026-01-29 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
WO-2002046170-A2 ANILINOPYRIMIDINE DERIVATIVES AS JNK PATHWAY INHIBITORS AND COMPOSITIONS AND METHODS RELATED THERETO SIGNAL PHARMACEUTICALS, INC. (US) 2002-06-13 WO claimed
WO-2002046171-A2 ANILINOPYRIMIDINE DERIVATIVES AS IKK INHIBITORS AND COMPOSITIONS AND METHODS RELATED THERETO SIGNAL PHARMACEUTICALS, INC. (US) 2002-06-13 WO claimed
US-20010049349-A1 Antioxidant enhancement of therapy for hyperproliferative conditions CRABTREE ACQUISITION CO, LLC 2001-12-06 US claimed
WO-2001032154-A2 USE OF TREOSULFAN FOR PATIENT CONDITIONING BEFORE BONE MARROW OR BLOOD STEM CELL TRANSPLANTATION Medac Gesellschaft für klinische Spezialpräparate mbH (DE) 2001-05-10 WO claimed
WO-2000045842-A2 METHODS FOR HUMAN ALLOGRAFTING THE GENERAL HOSPITAL CORPORATION (US) 2000-08-10 WO claimed
CN-1261803-A Antioxidant enhancement of therapy for hyperproliferative conditions ATHEROGENICS INC (US) 2000-08-02 CN claimed
EP-1019034-A2 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS Atherogenics, Inc. (US) 2000-07-19 EP claimed
WO-2000020022-A1 METHODS FOR THE TREATMENT OF CANCER USING CYTOKINES IN COMBINATION WITH LOW LEVEL DOSES OF CHEMOTHERAPY AND/OR RADIOTHERAPY LT TECHNOLOGY COMPANY, LLC. (US) 2000-04-13 WO claimed
WO-1999001118-A9 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS ATHEROGENICS INC (US) 1999-05-20 WO claimed
WO-1999001118-A2 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS ATHEROGENICS, INC. (US) 1999-01-14 WO claimed