Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL8146359

N#Cc1cccc(C[C@@H](NCc2cccc(Cn3c(=O)n(-c4ccccc4)n(-c4ccccc4)c3=O)c2)C(N)=O)c1.O=C(O)C(F)(F)F

nearest known ligand 0.39

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.39
SLC2A1 P11166 1/20 0.39
GPR6 P46095 1/20 0.38
GRIN1 Q05586 2/20 0.38
GRIN2B Q13224 2/20 0.38
KLKB1 P03952 2/20 0.37
F11 P03951 1/20 0.37
KLK1 P06870 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CCR2 P41597 1/20 0.36
FAAH O00519 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
CFTR P13569 1/20 0.35
MEP1B Q16820 2/20 0.35
VNN1 O95497 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
GPR34 Q9UPC5 1/20 0.35
FOLH1 Q04609 1/20 0.35
GNRHR P30968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8137836 0.81 TACR1 (0.41) SLC2A1GPR6GRIN1GRIN2BKLKB1
Trifluoroacetic Acid SCHEMBL8138243 0.79 F2 (0.42) SLC2A1KLKB1F11KLK1GPR34
Trifluoroacetic Acid SCHEMBL9287698 0.79 F11 (0.35) SLC2A1GPR6GRIN1GRIN2BKLKB1
SCHEMBL8126612 0.76 FEN1 (0.52) FEN1GRIN1GRIN2BL3MBTL1CCR2
SCHEMBL8143580 0.74 FEN1 (0.39) FEN1KLKB1KLK1CCR2MEP1B
SCHEMBL8153256 0.73 FEN1 (0.41) FEN1KLKB1KLK1CCR2FAAH
SCHEMBL8530291 0.72 ERCC1 (0.45) KLKB1KLK1DPP7MEP1BVNN1
SCHEMBL7354251 0.70 EPHX1 (0.46) DPP7MEP1BVNN1FOLH1
SCHEMBL7354256 0.70 EPHX1 (0.46) DPP7MEP1BVNN1FOLH1
Trifluoroacetic Acid SCHEMBL3488528 0.69 VNN1 (0.48) SLC2A1GPR6DPP7MEP1BVNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed
US-5616620-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-04-01 US disclosed
EP-0680469-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1995-11-08 EP disclosed
WO-1994017035-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME DR. KARL THOMAE GMBH (DE) 1994-08-04 WO disclosed