SCHEMBL8147398

SCHEMBL8147398

COc1cc2c(cc1OC)-c1cc(N)nc(=O)n1CC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.67
HSD17B10 Q99714 8/20 0.67
TSHR P16473 8/20 0.67
MAPK1 P28482 8/20 0.67
HPGD P15428 6/20 0.67
LMNA P02545 3/20 0.67
MAPT P10636 3/20 0.67
KDM4E B2RXH2 11/20 0.65
POLB P06746 4/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
KMT2A Q03164 3/20 0.61
MEN1 O00255 1/20 0.61
JAK2 O60674 1/20 0.61
GPR84 Q9NQS5 3/20 0.60
USP2 O75604 2/20 0.60
HTT P42858 1/20 0.60
HK1 P19367 1/20 0.60
HKDC1 Q2TB90 1/20 0.60
ALOX15 P16050 1/20 0.60
GLA P06280 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14137941 0.85 ALDH1A1 (0.68) ALDH1A1HSD17B10TSHRMAPK1HPGD
SCHEMBL30640051 0.84 ALDH1A1 (0.67) ALDH1A1HSD17B10TSHRMAPK1HPGD
SCHEMBL5117237 0.84 ALDH1A1 (0.67) ALDH1A1HSD17B10TSHRMAPK1HPGD
SCHEMBL4458547 0.82 GPR84 (0.62) ALDH1A1HSD17B10TSHRMAPK1HPGD
Iodide SCHEMBL10907785 0.81 ALDH1A1 (0.63) ALDH1A1HSD17B10TSHRMAPK1HPGD
SCHEMBL10907555 0.80 GPR84 (0.78) ALDH1A1HSD17B10TSHRMAPK1HPGD
Buquiterine SCHEMBL29387250 0.79 KDM4E (0.72) ALDH1A1HSD17B10TSHRMAPK1HPGD
SCHEMBL30798841 0.79 ALDH1A1 (0.60) ALDH1A1HSD17B10TSHRMAPK1HPGD
Buquiterine SCHEMBL2109704 0.79 KDM4E (0.72) ALDH1A1HSD17B10TSHRMAPK1HPGD
SCHEMBL7248968 0.78 GPR84 (0.79) ALDH1A1HSD17B10TSHRMAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973773-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 2000-01-26 EP disclosed
WO-1998045293-A1 PYRIMIDO-ISOQUINOLINE COMPOUNDS WITH ANTICONVULSIVE ACTION SMITHKLINE BEECHAM PLC (GB) 1998-10-15 WO disclosed