SCHEMBL8147495

SCHEMBL8147495

CCCCCCc1cc2c(cc1C#Cc1ccc(OC(C)=O)cn1)C(CC)(CC)CCO2

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.35
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
ACACB O00763 3/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
TSHR P16473 1/20 0.31
FPR1 P21462 1/20 0.31
APP P05067 1/20 0.30
BACE1 P56817 1/20 0.30
RXRA P19793 1/20 0.30
HNF4A P41235 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8661565 0.93 KMT2A (0.31) PTGDR2MEN1ALDH1A1KMT2A
SCHEMBL7652366 0.86 KMT2A (0.44) PTGDR2TSHRRXRAHNF4AMEN1
SCHEMBL7653907 0.85 ALDH1A1 (0.34) PTGDR2ALDH1A1
SCHEMBL8662212 0.84 CYP3A4 (0.38) ALOX5PTGDR2ACACBPPARGPPARA
SCHEMBL8661568 0.84 CYP3A4 (0.33) PTGDR2ACACBPPARGPPARAKMT2A
SCHEMBL8663351 0.84 KMT2A (0.31) ACACBRXRAHNF4AALDH1A1KMT2A
SCHEMBL7652859 0.83 CYP3A4 (0.33) PTGDR2ACACBPPARGPPARAKMT2A
SCHEMBL8659444 0.82
SCHEMBL8672856 0.82 ALOX5 (0.32) ALOX5
SCHEMBL8663068 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090826-A Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity ALLERGAN SALES, INC. (US) 2000-07-18 US disclosed