SCHEMBL8147641

SCHEMBL8147641

CC(C(=O)O)c1nc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(F)c(F)c2)o1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.48
PTGS1 P23219 12/20 0.48
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
SOS1 Q07889 1/20 0.39
LDHA P00338 1/20 0.38
LDHB P07195 1/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA12 O43570 1/20 0.37
CA4 P22748 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7504997 0.88 PTGS2 (0.63) PTGS2PTGS1CA1CA2CA12
SCHEMBL6002469 0.85 PTGS2 (0.50) PTGS2PTGS1CA1CA2CA12
SCHEMBL5823861 0.85 PTGS2 (0.50) PTGS2PTGS1CA1CA2CA12
SCHEMBL8619059 0.78 NR4A2 (0.53) PTGS2PTGS1SOS1LDHALDHB
SCHEMBL5732860 0.78 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL5732399 0.78 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL6000527 0.77 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6000535 0.75 PTGS2 (0.63) PTGS2PTGS1
SCHEMBL8145237 0.75 PTGS2 (0.51) PTGS2PTGS1SOS1CA1CA2
SCHEMBL27638570 0.74 CYP1A2 (0.43) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090834-A ANALGESICS; RHEUMATIC DISORDERS; SKIN DISORDERS; GASTROINTESTINAL DISORDERS G.D. SEARLE & CO. (US) 2000-07-18 US disclosed
WO-1996036617-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-11-21 WO disclosed