SCHEMBL8148282

SCHEMBL8148282

Oc1nccc2cc(OC3CC3)ccc12

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 15/20 0.57
ROCK2 O75116 3/20 0.49
KCNH2 Q12809 2/20 0.49
IKBKB O14920 1/20 0.43
PRKACA P17612 1/20 0.42
PRKCD Q05655 1/20 0.42
PRKG1 Q13976 1/20 0.42
PKN1 Q16512 1/20 0.42
PKN2 Q16513 1/20 0.42
AAK1 Q2M2I8 1/20 0.42
CDC42BPA Q5VT25 1/20 0.42
Q6ZSR9 Q6ZSR9 1/20 0.42
BMP2K Q9NSY1 1/20 0.42
CDC42BPB Q9Y5S2 1/20 0.42
PRKCZ Q05513 1/20 0.40
ABL1 P00519 2/20 0.39
FDPS P14324 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12211290 0.93 ROCK1 (0.54) ROCK1ROCK2KCNH2IKBKBPRKACA
Sar-407899 Free Base SCHEMBL8934240 0.90 ROCK1 (0.72) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL14981035 0.88 ROCK1 (0.49) ROCK1ROCK2KCNH2
SCHEMBL8939214 0.85 ROCK1 (0.54) ROCK1ROCK2KCNH2
SCHEMBL8939223 0.82 HRH3 (0.53) ROCK1ROCK2KCNH2
SCHEMBL3372945 0.81 ROCK1 (0.57) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL8939216 0.81 MAOA (0.53) ROCK1ROCK2KCNH2
SCHEMBL13763597 0.79 ROCK1 (0.54) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL13763659 0.78 ROCK1 (0.53) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL8271650 0.78 ALDH1A1 (0.46) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009005677-A2 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2009-01-08 WO disclosed