SCHEMBL8148997

SCHEMBL8148997

COc1ccc(F)c(Oc2cc(OC)ccc2F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.54
CA1 P00915 2/20 0.54
CA2 P00918 2/20 0.54
CA7 P43166 2/20 0.54
CA9 Q16790 2/20 0.54
CA14 Q9ULX7 2/20 0.54
CYP1A2 P05177 6/20 0.47
CYP1A1 P04798 5/20 0.47
CYP1B1 Q16678 5/20 0.47
ALDH1A1 P00352 4/20 0.47
CYP3A4 P08684 2/20 0.47
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
GAA P10253 1/20 0.43
CYP2A6 P11509 2/20 0.42
CYP2E1 P05181 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2219799 0.88 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL27274613 0.86 LTA4H (0.55) CA12CA1CA2CA7CA9
SCHEMBL7236023 0.81 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL1286402 0.81 CA12 (0.48) CA12CA1CA2CA7CA9
SCHEMBL12093386 0.79 HTT (0.47) CA12CA1CA2CA7CA9
SCHEMBL19862416 0.79 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL12093570 0.79 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL27891364 0.79 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL29835286 0.79 ALDH1A1 (0.46) CA12CA1CA2CA7CA9
SCHEMBL26919161 0.79 ALDH1A1 (0.46) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686145-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-01-26 EP disclosed
US-5883129-A Hydroxylated anthranilic acid derivatives ASTRA AKTIEBOLAG (SE) 1999-03-16 US disclosed
US-5523475-A New compounds AKTIEBOLAGET ASTRA (SE) 1996-06-04 US disclosed
CN-1121345-A New compounds ASTRA AB (SE) 1996-04-24 CN disclosed
EP-0686145-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1995-12-13 EP disclosed
WO-1994019316-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1994-09-01 WO disclosed