SCHEMBL8150163

SCHEMBL8150163

Clc1cccc2c1N=N[N]2

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.35
CYP2A6 P11509 2/20 0.35
TSHR P16473 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL792902 0.73 ALDH1A1 (0.36) CYP1A2TSHRALDH1A1LMNAKMT2A
SCHEMBL10588380 0.73
SCHEMBL5601076 0.66 NPC1 (0.37) CYP1A2TSHRALDH1A1
SCHEMBL5602519 0.65 ENPP1 (0.34) TSHRALDH1A1MEN1KMT2ATDP1
SCHEMBL5600567 0.65 NOS1 (0.38)
SCHEMBL4821733 0.64 CYP1A2 (0.35) CYP1A2CYP2A6TSHRALDH1A1LMNA
SCHEMBL5600295 0.63 NOS1 (0.39)
Water SCHEMBL20742739 0.62 MAPT (0.33)
SCHEMBL2294957 0.62 MAPT (0.33)
SCHEMBL10469489 0.60 MAPK13 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3400223-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES Syngenta Participations AG (CH) 2018-11-14 EP disclosed
WO-2017118689-A1 MICROBIOCIDAL OXADIAZOLE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2017-07-13 WO disclosed
US-6130220-A ENZYME INHIBITORS SYNTEX (USA) INC. (US) 2000-10-10 US disclosed
US-4242507-A Sulfonic acid esters FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-12-30 US disclosed