SCHEMBL8150807

SCHEMBL8150807

Cc1c2cc(C(=O)NCCCl)[nH]c2cc2c1sc1ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
POLB P06746 1/20 0.41
KDM4E B2RXH2 7/20 0.41
DRD2 P14416 2/20 0.40
DRD3 P35462 1/20 0.40
ALDH1A1 P00352 5/20 0.39
HTT P42858 2/20 0.39
HPGD P15428 2/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTR2C P28335 1/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HSD17B10 Q99714 1/20 0.37
RHEB Q15382 1/20 0.37
TNKS O95271 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8148345 0.90 ALDH1A1 (0.48) NPC1RAB9APOLBKDM4EDRD2
SCHEMBL8154275 0.80 ALDH1A1 (0.50) POLBKDM4EALDH1A1HTTHPGD
SCHEMBL8150334 0.77 ALDH1A1 (0.50) NPC1RAB9AKDM4EALDH1A1HTT
SCHEMBL8516897 0.75 KDM4E (0.33) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8150808 0.71 TNKS (0.42) RAB9APOLBKDM4EALDH1A1HTT
SCHEMBL8604346 0.70 ESR1 (0.39) NPC1RAB9APOLBKDM4EALDH1A1
SCHEMBL27015810 0.69 KDM4E (0.72) KDM4EDRD2DRD3ALDH1A1MAPK1
SCHEMBL14133855 0.65 MAPT (0.58) RAB9APOLBKDM4EALDH1A1HPGD
SCHEMBL8909780 0.65 KDM4E (0.48) NPC1RAB9AKDM4EDRD2DRD3
SCHEMBL22045050 0.64 TNKS (0.55) RAB9AKDM4EALDH1A1HTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999045926-A1 CONDENSED HETEROCYCLIC COMPOUNDS AS ANTI-INFLAMMATORY AND IMMUNOMODULATORY AGENTS UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1999-09-16 WO claimed
US-5852204-A Pyrrolo 3,2-b-!-carbazoles and 1H 1!benzothieno 2,3-f! indoles having anti-tumor activity UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1998-12-22 US claimed
EP-0741729-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1996-11-13 EP claimed
WO-1995021170-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-10 WO claimed
US-6013807-A Antitumor tetracyclic compounds UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 2000-01-11 US disclosed
US-5852204-A Pyrrolo 3,2-b-!-carbazoles and 1H 1!benzothieno 2,3-f! indoles having anti-tumor activity UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1998-12-22 US disclosed
US-5770598-A ANTITUMOR AGENTS; REACTING WITH CARBONYL DIIMIDAZOLE AND AMIDOXIMES UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1998-06-23 US disclosed
EP-0741729-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1996-11-13 EP disclosed
WO-1995021170-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-10 WO disclosed