SCHEMBL8516897

SCHEMBL8516897

CC1=C(C(=O)NCCCN)N=c2cc3c(c(C)c21)=Nc1ccccc1-3.Cc1c2cc(C(=O)NCCCl)[nH]c2cc2c1sc1ccccc12.Cc1c2cc(C(=O)NCCO)[nH]c2cc2c1sc1ccccc12

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 1/20 0.33
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8363292 0.97 KDM4E (0.35) KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9048962 0.79 PDCD1 (0.34) KDM4EALDH1A1HPGD
SCHEMBL8146941 0.78 GRIN1 (0.39) KDM4EHSD17B10HPGD
SCHEMBL8154329 0.76 KMT2A (0.31) KDM4EALDH1A1
SCHEMBL8147658 0.75 PDCD1 (0.37) KDM4EALDH1A1HPGD
SCHEMBL8150807 0.75 NPC1 (0.41) KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL8148345 0.74 ALDH1A1 (0.48) KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL8149445 0.74 TERT (0.36) KDM4E
SCHEMBL8365424 0.71
SCHEMBL8536552 0.67 GAA (0.32) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999045926-A1 CONDENSED HETEROCYCLIC COMPOUNDS AS ANTI-INFLAMMATORY AND IMMUNOMODULATORY AGENTS UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1999-09-16 WO disclosed