SCHEMBL8154178

SCHEMBL8154178

O=c1[nH]nc(Cc2ccc(Br)cc2)c2ccccc12

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.77
PARP1 P09874 3/20 0.77
LMNA P02545 1/20 0.73
ENPP1 P22413 2/20 0.61
TSHR P16473 2/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
PRMT5 O14744 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL863462 0.87 AR (1.00) ARPARP1LMNAENPP1TSHR
SCHEMBL2536051 0.85 PARP1 (0.72) ARPARP1LMNAENPP1TSHR
SCHEMBL12955526 0.84 AR (0.77) ARPARP1LMNAENPP1TSHR
SCHEMBL12955544 0.84 AR (0.77) ARPARP1LMNAENPP1TSHR
SCHEMBL7122967 0.84 AR (0.77) ARPARP1LMNAENPP1TSHR
SCHEMBL12955341 0.84 AR (0.77) ARPARP1LMNAENPP1TSHR
SCHEMBL29349943 0.84 LMNA (1.00) ARPARP1LMNAENPP1TSHR
SCHEMBL1789242 0.84 LMNA (1.00) ARPARP1LMNAENPP1TSHR
SCHEMBL4573019 0.84 PARP1 (0.70) ARPARP1LMNATSHRCYP3A4
SCHEMBL17825199 0.84 PARP1 (0.71) ARPARP1LMNAENPP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1330442-B1 PHTHALAZINONE DERIVATIVES KUDOS PHARM LTD (GB) 2011-01-19 EP disclosed
US-7750006-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2010-07-06 US disclosed
US-20080280910-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2008-11-13 US disclosed
US-20080280910-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2008-11-13 US disclosed
WO-2008114023-A2 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2008-09-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080280910-A1 PHTHALAZINONE DERIVATIVES H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, SDHA, NCOA4 AR 392/4885PARP1 3512/4885LMNA 1413/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.