SCHEMBL8154358

SCHEMBL8154358

C=C(c1ccc(C#Cc2ccccc2)cc1)N1CCN(c2ccccc2F)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
ALOX15 P16050 1/20 0.53
KMT2A Q03164 5/20 0.48
SMN1; SMN2 Q16637 5/20 0.48
ALDH1A1 P00352 4/20 0.48
MEN1 O00255 4/20 0.48
MAPK1 P28482 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TSHR P16473 2/20 0.48
GAA P10253 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
HTT P42858 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3638379 0.84 KDM4E (0.77) KDM4EALOX15KMT2ASMN1; SMN2ALDH1A1
SCHEMBL8160906 0.84 ADRA2C (0.44) KDM4EALOX15KMT2ASMN1; SMN2ALDH1A1
SCHEMBL8163764 0.82 GRM5 (0.48) KMT2AALDH1A1MEN1MAPK1TSHR
SCHEMBL8162119 0.77 GRM5 (0.68) KDM4EKMT2AALDH1A1TSHRMAPT
SCHEMBL8167707 0.75 MAPK1 (0.57) KDM4EKMT2AALDH1A1MEN1MAPK1
SCHEMBL8161908 0.75 SIGMAR1 (0.46) ALDH1A1HSD17B10TSHRUSP2GRM5
SCHEMBL8171420 0.74 GRM5 (0.49) GRM5
SCHEMBL8163323 0.73 GRM5 (0.69) KDM4EKMT2ASMN1; SMN2MEN1GAA
SCHEMBL8157655 0.73 GRM5 (0.44) ALOX15KMT2ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL8160767 0.72 GRM5 (0.52) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed