SCHEMBL8161908

SCHEMBL8161908

C=C(c1ccc(C#Cc2ccccc2)cc1)N1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.46
GRM5 P41594 7/20 0.46
POLB P06746 1/20 0.39
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CETP P11597 1/20 0.38
APP P05067 1/20 0.38
OPRD1 P41143 2/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
ADRB1 P08588 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
ABCC1 P33527 1/20 0.37
EGFR P00533 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14666451 0.85 SIGMAR1 (0.61) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL3640363 0.81 SIGMAR1 (0.73) SIGMAR1GRM5
SCHEMBL8162119 0.81 GRM5 (0.68) GRM5POLBALDH1A1TSHR
SCHEMBL8163323 0.80 GRM5 (0.69) GRM5APP
SCHEMBL8163764 0.80 GRM5 (0.48) GRM5POLBUSP2ALDH1A1TSHR
SCHEMBL8161856 0.80 GRM5 (0.50) GRM5
SCHEMBL16383677 0.78 LTA4H (0.47) SIGMAR1POLBUSP2ALDH1A1TSHR
SCHEMBL8154259 0.78 GRM3 (0.52) GRM5POLBALDH1A1
SCHEMBL8171420 0.78 GRM5 (0.49) GRM5
SCHEMBL8166622 0.77 CA12 (0.45) SIGMAR1GRM5POLBALDH1A1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed