SCHEMBL8154758

SCHEMBL8154758

CC(C)c1ccc(CC2=NCCN2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 6/20 1.00
HTR1B P28222 5/20 1.00
ADRA2A P08913 3/20 0.62
ADRA2B P18089 3/20 0.62
ADRA2C P18825 3/20 0.62
ADRA1D P25100 3/20 0.62
ADRA1A P35348 3/20 0.62
ADRA1B P35368 3/20 0.62
TAAR1 Q96RJ0 4/20 0.62
CYP2D6 P10635 2/20 0.62
LMNA P02545 1/20 0.62
CYP1A2 P05177 1/20 0.62
TSHR P16473 1/20 0.62
RAD52 P43351 1/20 0.57
NFKB1 P19838 1/20 0.56
NISCH Q9Y2I1 4/20 0.54
PTGIR P43119 1/20 0.54
MAOA P21397 3/20 0.50
MAOB P27338 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8146825 0.98 HTR1D (0.97) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL953972 0.81 RAD52 (0.82) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL2869241 0.81 HTR1D (0.69) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL4037274 0.79 HTR1D (0.71) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL9393147 0.77 HTR1D (0.69) HTR1DHTR1BADRA2AADRA2BADRA2C
Tolazoline SCHEMBL34961 0.77 TAAR1 (1.00) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL10846015 0.77 TAAR1 (0.72) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL9575262 0.77 PTGIR (0.83) HTR1DHTR1BADRA2AADRA2BADRA2C
SCHEMBL7986545 0.77 HTR1D (1.00) HTR1DHTR1BADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL7983686 0.75 HTR1D (0.97) HTR1DHTR1BADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048862-A Benzylamidine derivatives with serotonin receptor binding activity VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-04-11 US claimed
US-6048862-A Benzylamidine derivatives with serotonin receptor binding activity VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-04-11 US disclosed
US-5969137-A TREATMENT OF NERVOUS SYSTEM DISORDERS VIRGINIA COMMONWEALTH UNIVERSITY (US) 1999-10-19 US disclosed