SCHEMBL8159015

SCHEMBL8159015

CCOC(=Cc1cccc(CC)c1)C(=O)c1ccc(OCC)c(OCC)c1OCC

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
HTT P42858 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 3/20 0.37
LMNA P02545 2/20 0.37
MAPK1 P28482 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
NR1H4 Q96RI1 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GLO1 Q04760 1/20 0.34
AKR1C3 P42330 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8159554 0.92 HTT (0.38) KMT2AHTTALDH1A1KDM4ELMNA
SCHEMBL8160025 0.86 AKR1C3 (0.37) ALDH1A1KDM4EMAPK1L3MBTL1TSHR
SCHEMBL8153179 0.85 ABCB1 (0.42) KMT2AHTTKDM4ELMNAL3MBTL1
SCHEMBL8159064 0.85 PTGES (0.39) ALDH1A1LMNAMAPK1L3MBTL1TSHR
SCHEMBL8159445 0.84 PTPN11 (0.39) KMT2AALDH1A1KDM4ELMNAMAPK1
SCHEMBL8152034 0.83 PTPN11 (0.41) KMT2AALDH1A1KDM4ELMNAMAPK1
SCHEMBL8146381 0.79 MEN1 (0.50) KMT2AHTTLMNAMAPK1L3MBTL1
SCHEMBL8146380 0.79 MEN1 (0.50) KMT2AHTTLMNAMAPK1L3MBTL1
SCHEMBL8158807 0.78 ALDH1A1 (0.38) KMT2AALDH1A1KDM4ELMNAMAPK1
SCHEMBL8154299 0.77 ALOX5 (0.41) KMT2AALDH1A1LMNAMAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996432-A2 BIOLOGICALLY ACTIVE 1,3-BIS-AROMATIC-PROP-2-EN-1-ONES, 1,3-BIS-AROMATIC-PROPAN-1-ONES, AND 1,3-BIS-AROMATIC-PROP-2-YN-1-ONES STATENS SERUMINSTITUT (DK) 2000-05-03 EP claimed
WO-1999000114-A2 BIOLOGICALLY ACTIVE 1,3-BIS-AROMATIC-PROP-2-EN-1-ONES, 1,3-BIS-AROMATIC-PROPAN-1-ONES, AND 1,3-BIS-AROMATIC-PROP-2-YN-1-ONES STATENS SERUM INSTITUT (DK) 1999-01-07 WO claimed