SCHEMBL8159949

SCHEMBL8159949

CN(C)CC[C@H]1Cc2ccccc2[C@H]1O

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.53
HRH1 P35367 4/20 0.53
CDK8 P49336 1/20 0.48
CDK5 Q00535 1/20 0.48
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
HTR2C P28335 2/20 0.39
DRD2 P14416 1/20 0.39
ADRA1A P35348 1/20 0.39
BLM P54132 1/20 0.38
TSHR P16473 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
OPRM1 P35372 1/20 0.36
HTR2B P41595 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6268863 1.00 HTR2A (0.53) HTR2AHRH1CDK8CDK5SLC6A2
SCHEMBL9334169 1.00 HTR2A (0.53) HTR2AHRH1CDK8CDK5SLC6A2
SCHEMBL7306430 0.84 SLC6A2 (0.38) HTR2AHRH1CDK8CDK5SLC6A2
SCHEMBL8152258 0.83 SLC6A2 (0.54) HTR2AHRH1SLC6A2SLC6A4HTR2C
SCHEMBL8152263 0.83 SLC6A2 (0.54) HTR2AHRH1SLC6A2SLC6A4HTR2C
SCHEMBL8152267 0.83 SLC6A2 (0.54) HTR2AHRH1SLC6A2SLC6A4HTR2C
SCHEMBL8158561 0.83 SLC6A2 (0.54) HTR2AHRH1SLC6A2SLC6A4HTR2C
SCHEMBL12362873 0.83 SLC6A2 (0.54) HTR2AHRH1SLC6A2SLC6A4HTR2C
SCHEMBL9422155 0.81 OPRM1 (0.42) BLMTSHRSIGMAR1OPRM1
SCHEMBL11551882 0.80 HTR2A (0.51) HTR2AHRH1CDK8CDK5SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000005206-A1 ARYLPIPERAZINE DERIVATIVES USEFUL AS URO-SELECTIVE ALPHA-1-ADRENOCEPTOR BLOCKERS RANBAXY LABORATORIES LIMITED (US) 2000-02-03 WO claimed
EP-0303961-B1 Novel antidepressants MERRELL DOW PHARMA (US) 1994-04-13 EP disclosed