SCHEMBL8160809

SCHEMBL8160809

COc1ccc(CCCCBr)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.54
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
ADRA1A P35348 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
ESR1 P03372 1/20 0.43
CYP19A1 P11511 1/20 0.43
ESR2 Q92731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81884 0.95 APLNR (0.56) APLNRCA12CA1CA2CA7
SCHEMBL30502829 0.87 APLNR (0.59) APLNRCA12CA1CA2CA7
SCHEMBL11538133 0.87 APLNR (0.59) APLNRCA12CA1CA2CA7
SCHEMBL30107392 0.87 APLNR (0.63) APLNRCA12CA1CA2CA7
SCHEMBL23203396 0.85 ADRA1A (0.60) CA12CA1CA2CA7CA9
SCHEMBL9551466 0.85 ADRA1A (0.60) CA12CA1CA2CA7CA9
SCHEMBL1155658 0.85 ADRA1A (0.60) CA12CA1CA2CA7CA9
SCHEMBL7267199 0.85 ADRA1A (0.60) CA12CA1CA2CA7CA9
SCHEMBL22939735 0.84 APLNR (0.56) APLNRHTR2AALDH1A1
SCHEMBL1171776 0.83 MEN1 (0.56) APLNRHTR2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686145-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-01-26 EP disclosed
US-5883129-A Hydroxylated anthranilic acid derivatives ASTRA AKTIEBOLAG (SE) 1999-03-16 US disclosed
US-5523475-A New compounds AKTIEBOLAGET ASTRA (SE) 1996-06-04 US disclosed
EP-0686145-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1995-12-13 EP disclosed
WO-1994019316-A1 NEW COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1994-09-01 WO disclosed