SCHEMBL8162675

SCHEMBL8162675

O=C1c2cc[c]cc2CCc2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.61
MAOA P21397 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
MAOB P27338 3/20 0.45
BCHE P06276 1/20 0.42
MAPK14 Q16539 2/20 0.42
AKR1B1 P15121 1/20 0.42
CYP2A6 P11509 1/20 0.41
MIF P14174 7/20 0.41
CYP19A1 P11511 2/20 0.41
PKM P14618 1/20 0.41
CYP11B2 P19099 1/20 0.41
MAPK1 P28482 1/20 0.41
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8174906 0.89 CES1 (0.61) CES1MAOAL3MBTL1TDP1MAOB
SCHEMBL476341 0.88 CES1 (0.46) CES1MAOAL3MBTL1TDP1MAOB
SCHEMBL29408351 0.82 CES1 (0.90) CES1MAOAL3MBTL1TDP1MAOB
SCHEMBL44496 0.82 CES1 (0.90) CES1MAOAL3MBTL1TDP1MAOB
SCHEMBL29437756 0.82 CES1 (0.90) CES1MAOAL3MBTL1TDP1MAOB
SCHEMBL27537566 0.78 MAOA (0.67) CES1MAOAL3MBTL1TDP1MAOB
SCHEMBL11251467 0.77 MAPT (0.53) CES1MAOATDP1MAOBMAPK14
SCHEMBL134194 0.77
SCHEMBL13712393 0.77 CES1 (1.00) CES1MAOAL3MBTL1TDP1MAOB
SCHEMBL4312831 0.76 CES1 (0.46) CES1MAOAL3MBTL1TDP1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043247-A A SUBSTITUTED ACRYLIC ACIDS FOR USE IN TREATMENT OF HUMAN AND ANIMAL DISORDERS, AND PURIFICATION OF PROTEINS OR GLYCOPROTEINS, AND TO THEIR USE IN DIAGNOSIS NOVO NORDISK A/S (DK) 2000-03-28 US claimed
US-6043247-A A SUBSTITUTED ACRYLIC ACIDS FOR USE IN TREATMENT OF HUMAN AND ANIMAL DISORDERS, AND PURIFICATION OF PROTEINS OR GLYCOPROTEINS, AND TO THEIR USE IN DIAGNOSIS NOVO NORDISK A/S (DK) 2000-03-28 US disclosed
WO-1997039748-A1 MODULATORS OF MOLECULES WITH PHOSPHOTYROSINE RECOGNITION UNITS NOVO NORDISK A/S (DK) 1997-10-30 WO disclosed