SCHEMBL8166235

SCHEMBL8166235

CCOC(=O)C(C(=O)OCC)C1CCc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.46
PPARA Q07869 1/20 0.46
TSHR P16473 1/20 0.44
FFAR1 O14842 2/20 0.43
DRD2 P14416 1/20 0.42
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
SLC6A2 P23975 3/20 0.41
SLC6A3 Q01959 3/20 0.41
SLC6A4 P31645 2/20 0.41
PIN1 Q13526 1/20 0.41
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
ALDH1A1 P00352 2/20 0.40
XBP1 P17861 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31758112 0.86 FFAR1 (0.41) PPARGPPARAFFAR1DRD2SLC6A2
SCHEMBL8301035 0.86 PPARG (0.43) PPARGPPARAFFAR1PIN1
SCHEMBL7961254 0.82 FFAR1 (0.49) PPARGPPARATSHRFFAR1MTNR1A
SCHEMBL7961253 0.82 FFAR1 (0.49) PPARGPPARATSHRFFAR1MTNR1A
SCHEMBL10742068 0.82 TSHR (0.43) TSHRFFAR1L3MBTL1PIN1HPGD
SCHEMBL13925659 0.82 ESR1 (0.56) PPARGPPARADRD2MTNR1AMTNR1B
SCHEMBL31072342 0.80 MTNR1B (0.52) MTNR1AMTNR1B
SCHEMBL10493642 0.79 ACE (0.42) PPARGPPARATSHRFFAR1MTNR1A
SCHEMBL10493648 0.79 ACE (0.42) PPARGPPARATSHRFFAR1MTNR1A
SCHEMBL31757646 0.79 MEN1 (0.39) PPARGPPARATSHRFFAR1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048852-A BACTERICIDES SMITHKLINE BEECHAM P.L.C. (GB) 2000-04-11 US disclosed
EP-0900197-A1 BETA-THIOPROPIONYL-AMINOACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1999-03-10 EP disclosed
WO-1997030027-A1 BETA-THIOPROPIONYL-AMINOACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1997-08-21 WO disclosed
US-4249021-A USEFUL AS DIURETIC AGENTS IN TREATMENT OF EDEMA; ALSO FOR TREATMENT OF HYPERTENSION MERCK & CO., INC. (US) 1981-02-03 US disclosed