SCHEMBL8168514

SCHEMBL8168514

CN(Cc1cc([N+](=O)[O-])ccc1N1CCCS1(=O)=O)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
MCOLN3 Q8TDD5 1/20 0.41
SMN1; SMN2 Q16637 6/20 0.39
MAPT P10636 3/20 0.37
GPR55 Q9Y2T6 1/20 0.37
GAA P10253 1/20 0.37
LMNA P02545 3/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8164427 0.97 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL18186410 0.85 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL16824953 0.85 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL16824841 0.84 ALDH1A1 (0.56) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL18186409 0.83 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL8163944 0.81 CALCA (0.38) ALDH1A1SMN1; SMN2MAPTGAAHTT
SCHEMBL16824900 0.80 SMN1; SMN2 (0.51) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL8164137 0.80 ALDH1A1 (0.37) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL8156882 0.80 HTT (0.46) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL18186205 0.79 LMNA (0.54) ALDH1A1CYP1A2CYP3A4CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008079836-A2 MACROCYCLIC FACTOR VIIA INHIBITORS USEFUL AS ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-07-03 WO disclosed