SCHEMBL8169549

SCHEMBL8169549

N=C(N)c1ccc(S(=O)(=O)c2cccc3cccnc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
ST14 Q9Y5Y6 1/20 0.53
TSHR P16473 1/20 0.48
HTT P42858 1/20 0.48
NAMPT P43490 3/20 0.47
GAA P10253 4/20 0.47
KDM4E B2RXH2 4/20 0.47
MAPT P10636 2/20 0.47
APOBEC3G Q9HC16 2/20 0.47
F2 P00734 2/20 0.46
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
ALDH1A1 P00352 3/20 0.44
KMT2A Q03164 1/20 0.44
CNR1 P21554 1/20 0.43
ALOX12 P18054 1/20 0.43
PARP1 P09874 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13241507 0.79 MAPK1 (0.62) MAPK1CA1CA2CA9TSHR
SCHEMBL7073865 0.79 MAPT (0.61) MAPK1CA1CA2CA9TSHR
SCHEMBL8162975 0.79 HTR6 (0.67) CA1CA2CA9ST14TSHR
SCHEMBL27429625 0.77 MAPT (0.60) MAPK1CA1CA2CA9TSHR
SCHEMBL30714537 0.73 L3MBTL1 (0.56) KDM4E
SCHEMBL4108638 0.73 MAPK1 (0.66) MAPK1CA1CA2CA9TSHR
Potassium Ion SCHEMBL31267534 0.73 MAPK1 (0.66) MAPK1CA1CA2CA9TSHR
SCHEMBL8170523 0.73 PKM (0.59) NAMPTKDM4EF2KMT2A
SCHEMBL7180056 0.72 MAPK1 (0.70) MAPK1CA1CA2CA9TSHR
SCHEMBL2459763 0.71 MAPK1 (0.68) MAPK1CA1CA2CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114328-A ANTICOAGULANTS; BLOOD DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-09-05 US disclosed
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed