SCHEMBL8175265

SCHEMBL8175265

Bc1ccc2c(c1)c(CC(=O)O)c(C(=O)N1CCNC(=O)C1)n2Cc1ccc(C(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
PTGES2 Q9H7Z7 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
LMNA P02545 2/20 0.36
TSHR P16473 2/20 0.36
CYP2C19 P33261 2/20 0.36
PMP22 Q01453 2/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.36
MAPK1 P28482 2/20 0.36
KMT2A Q03164 2/20 0.36
RGS12 O14924 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
NFKB1 P19838 1/20 0.36
GNAI1 P63096 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13931384 0.91 PTGS2 (0.42) PARP1PARP2PTGES2CYP1A2CYP3A4
SCHEMBL8181544 0.89 CYP1A2 (0.39) PTGES2CYP1A2CYP3A4CYP2C9LMNA
SCHEMBL8175786 0.86 KMT2A (0.41) PTGES2CYP1A2CYP3A4CYP2C9LMNA
SCHEMBL13931385 0.80 PTGS2 (0.44) PTGES2CYP1A2CYP3A4CYP2C9LMNA
SCHEMBL13931386 0.77 PTGS2 (0.46) PTGES2CYP1A2CYP3A4CYP2C9LMNA
SCHEMBL8181548 0.76 PPARG (0.40) PTGES2CYP1A2CYP3A4CYP2C9LMNA
SCHEMBL8179608 0.75 ATM (0.49) CYP1A2CYP3A4CYP2C9LMNATSHR
SCHEMBL8167668 0.75 PLA2G1B (0.43) CYP1A2CYP3A4CYP2C9LMNATSHR
SCHEMBL8165177 0.74 PPARG (0.47) MEN1KMT2AALDH1A1PTGDR2PTGES
SCHEMBL8171613 0.72 PPARG (0.50) PTGES2PLA2G2ATHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008100867-A2 NOVEL INHIBITORS HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2008-08-21 WO disclosed