SCHEMBL8175607

SCHEMBL8175607

c1ccc(C(c2ccccc2)N2CCN(C(c3ccccc3)c3ccccc3)CCN(C(c3ccccc3)c3ccccc3)CCN(C(c3ccccc3)c3ccccc3)CCN(C(c3ccccc3)c3ccccc3)CC2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.78
CYP2D6 P10635 3/20 0.78
CHRM2 P08172 2/20 0.78
ADRA2A P08913 2/20 0.78
CHRM1 P11229 2/20 0.78
DRD1 P21728 2/20 0.78
DRD3 P35462 2/20 0.78
SLC6A3 Q01959 2/20 0.78
KCNH2 Q12809 2/20 0.78
CHRM4 P08173 1/20 0.78
CHRM5 P08912 1/20 0.78
ADORA3 P0DMS8 1/20 0.78
CHRM3 P20309 1/20 0.78
ADRA1D P25100 1/20 0.78
HTR2A P28223 1/20 0.78
HTR2C P28335 1/20 0.78
HRH1 P35367 1/20 0.78
HTR2B P41595 1/20 0.78
KMT2A Q03164 5/20 0.71
MEN1 O00255 3/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8186671 1.00 OPRM1 (0.78) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL7977689 1.00 OPRM1 (0.78) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL3919536 1.00 OPRM1 (0.78) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL8176312 0.91 OPRM1 (0.67) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL7317034 0.91 OPRM1 (0.67) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL1502253 0.90 CYP2D6 (0.65) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL2054235 0.90 CYP2D6 (0.67) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL467087 0.89 OPRM1 (0.64) OPRM1CYP2D6CHRM2ADRA2ACHRM1
SCHEMBL16448455 0.89 OPRM1 (0.70) OPRM1CYP2D6CHRM2ADRA2ACHRM1
Cyclizine SCHEMBL4690 0.89 CYP2D6 (1.00) OPRM1CYP2D6CHRM2ADRA2ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048979-A CYCLOTETRAMERIZING, CLEAVAGE OF ARYLMETHYL GROUPS TO PREPARE CYCLEN AND DERIVATIVES NYCOMED SALUTAR, INC. (US) 2000-04-11 US disclosed