SCHEMBL8176753

SCHEMBL8176753

Cc1ccc(NC(=O)c2cn(Cc3ccccc3)cn2)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
MAPT P10636 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
HPGD P15428 1/20 0.54
KLKB1 P03952 2/20 0.53
NPSR1 Q6W5P4 1/20 0.52
RIPK1 Q13546 1/20 0.48
USP30 Q70CQ3 1/20 0.47
RBP4 P02753 1/20 0.46
KDR P35968 1/20 0.46
CNR1 P21554 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
HSP90AA1 P07900 1/20 0.46
NLRP3 Q96P20 1/20 0.46
TLR9 Q9NR96 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18377475 0.82 KLKB1 (0.56) KLKB1RIPK1USP30RBP4
SCHEMBL15965171 0.79 KLKB1 (0.47) KLKB1RBP4
SCHEMBL24094049 0.79 KLKB1 (0.55) KLKB1RIPK1USP30RBP4
SCHEMBL23432082 0.79 KLKB1 (0.53) MEN1KMT2AKLKB1RIPK1USP30
SCHEMBL19304343 0.78 ALDH1A1 (0.53) MAPTMEN1KMT2A
SCHEMBL31073512 0.78 MEN1 (0.56) MAPTMEN1KMT2AHPGDKLKB1
SCHEMBL16690901 0.78 RBP4 (0.54) NPC1RAB9ASMN1; SMN2KLKB1RIPK1
SCHEMBL3688462 0.77 KDM4C (0.57) NPC1RAB9AKLKB1RIPK1USP30
SCHEMBL18367381 0.77 CDK5 (0.53) SMN1; SMN2MEN1KMT2AKLKB1RIPK1
SCHEMBL24310642 0.75 KDM4C (0.52) NPC1RAB9AKLKB1RIPK1USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed