SCHEMBL8177809

SCHEMBL8177809

O=c1[nH]nc(S)n1-c1cccc(F)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
FAAH O00519 1/20 0.44
MGLL Q99685 1/20 0.44
NOTUM Q6P988 3/20 0.42
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
ALOX5 P09917 2/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KEAP1 Q14145 1/20 0.37
MDM2 Q00987 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8186274 0.80 ALDH1A1 (0.44) MGLLNOTUMALDH1A1POLB
SCHEMBL8178332 0.80 GSK3A (0.50) CYP1A2ALDH1A1GAAKMT2AMEN1
SCHEMBL8177807 0.79 NOTUM (0.41) CYP1A2NOTUMALDH1A1POLBSMN1; SMN2
SCHEMBL8177459 0.79 CYP1A2 (0.74) CYP1A2MGLLNOTUMALDH1A1POLB
SCHEMBL17537374 0.72 FAAH (0.59) CYP1A2FAAHMGLLNOTUMALDH1A1
SCHEMBL8185793 0.70 CYP1A2 (0.54) CYP1A2NOTUMALDH1A1POLBRAB9A
SCHEMBL8187626 0.70 CYP2C9 (0.74) CYP1A2GAAMAPT
SCHEMBL23931446 0.69 HTT (0.65) FAAHMGLLNOTUMALDH1A1POLB
SCHEMBL8177088 0.69 MAPK8 (0.53) NOTUMALDH1A1POLBGAAMAPT
SCHEMBL8187437 0.69 BRD9 (0.50) ALDH1A1POLBMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008118626-A9 INHIBITORS OF JNK AND METHODS FOR IDENTIFYING INHIBITORS OF JNK BURNHAM INST MEDICAL RESEARCH (US) 2008-12-18 WO disclosed
WO-2008118626-A2 INHIBITORS OF JNK AND METHODS FOR IDENTIFYING INHIBITORS OF JNK BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2008-10-02 WO disclosed