SCHEMBL8180271

SCHEMBL8180271

CCOC(=O)C1CCN(c2nc(NCc3ccccc3)c3cc([N+](=O)[O-])sc3n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 11/20 0.44
TCF7L2 Q9NQB0 11/20 0.44
CTSB P07858 1/20 0.44
MAPT P10636 4/20 0.44
TP53 P04637 1/20 0.43
HTT P42858 1/20 0.43
ALDH1A1 P00352 2/20 0.43
PTPN11 Q06124 1/20 0.42
GAA P10253 1/20 0.42
PDE5A O76074 1/20 0.42
HRH4 Q9H3N8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8184659 0.92 MAPT (0.45) CTSBMAPTTP53HTTALDH1A1
SCHEMBL8185688 0.92 CTNNB1 (0.46) CTNNB1TCF7L2MAPTTP53HTT
SCHEMBL8179215 0.89 ALDH1A1 (0.47) CTNNB1TCF7L2CTSBMAPTTP53
SCHEMBL8180789 0.89 PDE4A (0.47) CTNNB1TCF7L2MAPTPDE5AHRH4
SCHEMBL7017521 0.89 HRH4 (0.41) CTNNB1TCF7L2PDE5AHRH4
SCHEMBL8185685 0.89 ALDH1A1 (0.46) CTSBMAPTTP53HTTALDH1A1
SCHEMBL8179602 0.88 CTNNB1 (0.48) CTNNB1TCF7L2MAPTALDH1A1PTPN11
SCHEMBL8179254 0.88 ICAM1 (0.48) CTNNB1TCF7L2MAPTHTTALDH1A1
SCHEMBL8171152 0.87 PDE4A (0.53) CTNNB1TCF7L2MAPTHTTALDH1A1
SCHEMBL8184614 0.87 PDE4A (0.48) CTSBMAPTTP53HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed