SCHEMBL8181739

SCHEMBL8181739

COC(=O)c1ccc(C#C/C=C/c2ccccc2-c2ccncc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 1/20 0.40
DYRK1A Q13627 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SLC2A1 P11166 1/20 0.38
PTPN11 Q06124 1/20 0.38
EGFR P00533 1/20 0.38
CYP46A1 Q9Y6A2 1/20 0.38
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 4/20 0.37
MAPT P10636 3/20 0.37
NPC1 O15118 1/20 0.37
NFKB1 P19838 1/20 0.37
RAB9A P51151 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ROCK2 O75116 1/20 0.37
POLB P06746 2/20 0.37
HPGD P15428 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8175916 0.91 EGFR (0.46) PTPN11EGFRKDM4EALDH1A1MAPT
SCHEMBL8175983 0.89 SLC2A1 (0.48) KMT2ASLC2A1KDM4EALDH1A1MAPT
SCHEMBL8167327 0.88 TDP1 (0.46) PTPN11EGFRKDM4EALDH1A1MAPT
SCHEMBL8180152 0.88 CA1 (0.46) PTPN11EGFRKDM4EALDH1A1HPGD
SCHEMBL8167359 0.87 CA1 (0.47) MEN1KMT2AEGFRKDM4EMAPT
SCHEMBL8166934 0.87 SLC6A4 (0.48) PTPN11EGFRKDM4EALDH1A1MAPT
SCHEMBL8175487 0.87 EGFR (0.40) MEN1KMT2APTPN11EGFRMAPT
SCHEMBL8175144 0.87 SLC6A4 (0.48) MEN1KMT2APTPN11EGFRKDM4E
SCHEMBL7930817 0.86 RARB (0.41) ALDH1A1
SCHEMBL8175888 0.86 PTPN1 (0.38) KMT2APTPN11EGFRKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6150413-A TREATMENT OF DERMATOLOGICAL, RHEUMATIC, RESPIRATORY, CARDIOVASCULAR, BONE AND OPHTHALMOLOGICAL DISORDERS, AS WELL AS MAMMALIAN SKIN AND HAIR CONDITIONS; 4-(4-(BIPHENYL-2-YL)BUT-3-EN-1-YNYL)BENZOIC ACID, FOR EXAMPLE CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (FR) 2000-11-21 US disclosed