SCHEMBL8175144

SCHEMBL8175144

COC(=O)c1ccc(C#C/C=C/c2ccccc2-c2ccc(F)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48
PTGS1 P23219 1/20 0.46
KMT2A Q03164 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 2/20 0.40
MAPK1 P28482 2/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
EGFR P00533 1/20 0.40
ATM Q13315 1/20 0.40
PTPRC P08575 1/20 0.39
PTPRF P10586 1/20 0.39
PTPN1 P18031 1/20 0.39
CDC25B P30305 1/20 0.39
ALDH1A1 P00352 3/20 0.38
PTPN11 Q06124 1/20 0.38
ERN1 O75460 1/20 0.37
TUBB4A P04350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8175916 0.91 EGFR (0.46) NPC1RAB9AMAPTEGFRPTPRC
SCHEMBL8180152 0.90 CA1 (0.46) EGFRPTPRCPTPRFPTPN1CDC25B
SCHEMBL8167327 0.90 TDP1 (0.46) NPC1RAB9AMAPTEGFRATM
SCHEMBL8167359 0.89 CA1 (0.47) KMT2ANPC1RAB9AMEN1MAPT
SCHEMBL8166934 0.89 SLC6A4 (0.48) SLC6A4SLC6A3NPC1RAB9AMAPT
SCHEMBL8175487 0.89 EGFR (0.40) KMT2ARAB9AMEN1MAPTEGFR
SCHEMBL8175888 0.88 PTPN1 (0.38) SLC6A4SLC6A3KMT2AMAPTEGFR
SCHEMBL8181712 0.87 EGFR (0.39) KMT2ANPC1RAB9AMEN1MAPT
SCHEMBL8181739 0.87 RAF1 (0.40) KMT2ANPC1RAB9AMEN1MAPT
SCHEMBL7929309 0.86 BCL2L1 (0.45) SLC6A4SLC6A3KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6150413-A TREATMENT OF DERMATOLOGICAL, RHEUMATIC, RESPIRATORY, CARDIOVASCULAR, BONE AND OPHTHALMOLOGICAL DISORDERS, AS WELL AS MAMMALIAN SKIN AND HAIR CONDITIONS; 4-(4-(BIPHENYL-2-YL)BUT-3-EN-1-YNYL)BENZOIC ACID, FOR EXAMPLE CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (FR) 2000-11-21 US disclosed