SCHEMBL8182789

SCHEMBL8182789

COc1c(C(=O)c2ccc(F)cc2F)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.41
CES2 O00748 3/20 0.41
CES1 P23141 1/20 0.41
GPBAR1 Q8TDU6 1/20 0.36
SCN8A Q9UQD0 2/20 0.36
SCN10A Q9Y5Y9 2/20 0.36
HTT P42858 2/20 0.36
KDM4E B2RXH2 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KMT2A Q03164 1/20 0.36
TMPRSS4 Q9NRS4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8176045 0.85 CES2 (0.40) CES2CES1GPBAR1SCN8ASCN10A
SCHEMBL8168125 0.81 CES2 (0.40) CES2CES1GPBAR1SCN8ASCN10A
SCHEMBL8177263 0.79 SCN8A (0.46) MAPK14CES2CES1SCN8ASCN10A
SCHEMBL8168954 0.76 MAPK14 (0.46) MAPK14CES2CES1HTTKMT2A
SCHEMBL22114934 0.76 HSD17B10 (0.44) CES2KDM4ETMPRSS4
SCHEMBL8176775 0.75 CES2 (0.47) MAPK14CES2CES1HTTKMT2A
SCHEMBL12247362 0.75 CES2 (0.41) CES2HTTKMT2ATMPRSS4
SCHEMBL30343770 0.75 NOTUM (0.50) CES2KDM4ETMPRSS4
SCHEMBL8175847 0.74 SMO (0.43) RXFP1KMT2ATMPRSS4
SCHEMBL8182159 0.72 TMPRSS4 (0.49) MAPK14CES2CES1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000063176-A2 DISUBSTITUTED PYRIDINES AND PYRIMIDINES AS HERBICIDES AND FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 2000-10-26 WO disclosed