SCHEMBL8183644

SCHEMBL8183644

COc1cc(OC)c(C(=O)Nc2ccc3c(c2)CN(C)CC3)cc1Br

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.52
CYP3A4 P08684 1/20 0.52
ABCB1 P08183 2/20 0.49
ABCG2 Q9UNQ0 2/20 0.49
KMT2A Q03164 5/20 0.48
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
MEN1 O00255 4/20 0.48
MAPT P10636 2/20 0.47
TSHR P16473 2/20 0.47
MAPK1 P28482 2/20 0.47
TP53 P04637 1/20 0.47
ACHE P22303 1/20 0.45
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
SLC6A4 P31645 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
HTR2A P28223 1/20 0.45
KDM4E B2RXH2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7792074 0.85 ROCK2 (0.51) ROCK2CYP3A4KMT2ANPC1RAB9A
SCHEMBL6293939 0.85 ROCK2 (0.65) ROCK2CYP3A4ABCB1ABCG2KMT2A
SCHEMBL8185594 0.85 ALDH1A1 (0.59) ROCK2CYP3A4KMT2ANPC1RAB9A
Hydrochloric Acid SCHEMBL7792070 0.85 NPC1 (0.59) ROCK2CYP3A4KMT2ANPC1RAB9A
SCHEMBL7849356 0.84 ROCK2 (0.56) ROCK2CYP3A4ABCB1ABCG2NPC1
SCHEMBL8184565 0.83 KMT2A (0.58) ROCK2CYP3A4KMT2ANPC1RAB9A
SCHEMBL8130831 0.83 ROCK2 (0.52) ROCK2CYP3A4ABCB1ABCG2KMT2A
SCHEMBL8188782 0.83 ACHE (0.64) ROCK2CYP3A4NPC1RAB9AMAPT
SCHEMBL6293671 0.83 F10 (0.48) ROCK2CYP3A4ABCB1ABCG2NPC1
SCHEMBL8191620 0.83 ROCK2 (0.54) ROCK2CYP3A4KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6110934-A Substituted benzamide derivatives and their use as anticonvulsants SMITHKLINE BEECHAM P.L.C. (GB) 2000-08-29 US disclosed
EP-0906283-A1 SUBSTITUTED BENZAMIDE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1999-04-07 EP disclosed
WO-1997048683-A1 SUBSTITUTED BENZAMIDE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1997-12-24 WO disclosed