SCHEMBL8185074

SCHEMBL8185074

CCNc1nc(CC)ccc1C(=O)c1cccc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 5/20 0.41
ADCY8 P40145 1/20 0.40
ADCY1 Q08828 1/20 0.40
CYP3A4 P08684 3/20 0.40
PDE4B Q07343 2/20 0.40
CYP2C19 P33261 1/20 0.40
ADORA2A P29274 1/20 0.40
PARP1 P09874 1/20 0.39
CHRNA7 P36544 1/20 0.38
ERCC5 P28715 1/20 0.38
FEN1 P39748 1/20 0.38
GRM5 P41594 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6221826 0.88 GRM5 (0.45) VNN1ADORA2APARP1CHRNA7ERCC5
SCHEMBL6221038 0.86 MAPT (0.45) VNN1ADORA2AGRM5
SCHEMBL8198909 0.86 POLB (0.45) VNN1ADCY8ADCY1PARP1GRM5
SCHEMBL8198347 0.86 TSHR (0.41) ADCY8ADCY1CYP2C19PARP1GRM5
SCHEMBL8198559 0.84 CYP3A4 (0.44) VNN1ADCY8ADCY1CYP3A4PDE4B
SCHEMBL6226517 0.83 VNN1 (0.40) VNN1CYP3A4CYP2C19ADORA2ACHRNA7
SCHEMBL8197231 0.83 VNN1 (0.40) VNN1ADORA2ACHRNA7ERCC5FEN1
SCHEMBL8196200 0.82 MAPT (0.40) VNN1CYP2C19ERCC5FEN1GRM5
SCHEMBL8198616 0.82 ADORA1 (0.48) VNN1CYP2C19ADORA2AGRM5
SCHEMBL6221993 0.81 HPGD (0.40) VNN1CHRNA7GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136810-A DRUGS AS ENZYME INHIBITORS OF PHOSPHODIESTERASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0885894-A1 PYRIDO [2,3-D] PYRIMIDINE DERIVATIVES AND MEDICINAL COMPOSITIONS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-23 EP disclosed