SCHEMBL8198616

SCHEMBL8198616

CCNc1nc(-c2ccccc2)ccc1C(=O)c1cccc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.48
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
LMNA P02545 1/20 0.47
VNN1 O95497 3/20 0.44
ADORA2A P29274 3/20 0.42
GRM5 P41594 1/20 0.41
ALOX15 P16050 1/20 0.40
CNR2 P34972 1/20 0.40
NLRP3 Q96P20 1/20 0.40
PTGER4 P35408 1/20 0.40
RECQL P46063 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CNR1 P21554 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6221826 0.84 GRM5 (0.45) VNN1ADORA2AGRM5ALOX15ALDH1A1
SCHEMBL6221038 0.83 MAPT (0.45) VNN1ADORA2AGRM5ALDH1A1MAPT
SCHEMBL8185074 0.82 VNN1 (0.41) CYP2C19VNN1ADORA2AGRM5
SCHEMBL8193773 0.81 ALDH1A1 (0.41) KMT2AMEN1VNN1GRM5CNR2
SCHEMBL8197231 0.81 VNN1 (0.40) VNN1ADORA2AGRM5ALOX15ALDH1A1
SCHEMBL6226517 0.81 VNN1 (0.40) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8196200 0.80 MAPT (0.40) KMT2ACYP1A2CYP2C19NPSR1LMNA
SCHEMBL6221993 0.79 HPGD (0.40) KMT2AMEN1VNN1GRM5ALDH1A1
SCHEMBL8692622 0.77 MEN1 (0.48) KMT2AMEN1VNN1KDM4EALDH1A1
SCHEMBL20256974 0.75 LDHA (0.45) ADORA1KMT2AMEN1ADORA2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136810-A DRUGS AS ENZYME INHIBITORS OF PHOSPHODIESTERASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0885894-A1 PYRIDO [2,3-D] PYRIMIDINE DERIVATIVES AND MEDICINAL COMPOSITIONS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-23 EP disclosed