SCHEMBL8185136

SCHEMBL8185136

CCc1cc2c(NCCc3ccc4c(c3)OCCO4)nc(-c3ccc(C(=O)O)cc3)nc2s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 3/20 0.48
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 3/20 0.43
THRB P10828 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
HTT P42858 2/20 0.42
MAPT P10636 1/20 0.42
CNR2 P34972 1/20 0.40
P2RY12 Q9H244 3/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8181651 0.95 PRKCI (0.48) PRKCIALDH1A1KDM4EHSD17B10LMNA
SCHEMBL8178110 0.92 PRKCI (0.47) PRKCIALDH1A1KDM4EHSD17B10LMNA
SCHEMBL8180183 0.90 ALDH1A1 (0.43) ALDH1A1KDM4ELMNATHRBCYP1A2
SCHEMBL8171150 0.89 LMNA (0.43) ALDH1A1HSD17B10LMNATHRBCYP1A2
SCHEMBL8180756 0.88 LMNA (0.43) ALDH1A1LMNATHRBCYP1A2CYP3A4
SCHEMBL7609419 0.88 PRKCI (0.64) PRKCIALDH1A1KDM4EHSD17B10CNR2
SCHEMBL8184670 0.86 PRKCI (0.47) PRKCIALDH1A1KDM4EHSD17B10LMNA
SCHEMBL8181999 0.86 PDE5A (0.52) PRKCIALDH1A1KDM4EHSD17B10LMNA
SCHEMBL8179775 0.86 LMNA (0.41) ALDH1A1LMNATHRBCYP1A2CYP3A4
SCHEMBL8185149 0.85 PRKCI (0.55) PRKCIALDH1A1KDM4EHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed