SCHEMBL8185282

SCHEMBL8185282

O=CNCc1ccncn1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 1/20 0.42
ADH1B P00325 1/20 0.39
ADH1C P00326 1/20 0.39
ADH1A P07327 1/20 0.39
ADH7 P40394 1/20 0.39
NAMPT P43490 3/20 0.38
P2RX7 Q99572 1/20 0.38
HPGDS O60760 1/20 0.35
MAPK14 Q16539 1/20 0.34
HSP90AA1 P07900 1/20 0.34
CHRM4 P08173 1/20 0.33
PDE10A Q9Y233 1/20 0.33
OPRM1 P35372 1/20 0.33
SLC40A1 Q9NP59 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8191782 0.81 P2RX7 (0.36) KCNH3ADH1BADH1AADH7NAMPT
SCHEMBL18157948 0.81 KCNH3 (0.47) KCNH3NAMPTP2RX7HPGDSMAPK14
SCHEMBL13100189 0.74 KCNH3 (0.43) KCNH3NAMPTP2RX7HPGDSMAPK14
SCHEMBL348051 0.74 HSP90AA1 (0.35) KCNH3NAMPTP2RX7HSP90AA1
SCHEMBL29953667 0.74 HSP90AA1 (0.35) KCNH3NAMPTP2RX7HSP90AA1
SCHEMBL399162 0.74 SMN1; SMN2 (0.56) ADH1BADH1CADH1AADH7
SCHEMBL4661605 0.74
SCHEMBL10188167 0.74
SCHEMBL553439 0.74
SCHEMBL8185279 0.73 KCNH3 (0.42) KCNH3NAMPTP2RX7HPGDSMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1947101-A1 HYDRAZIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR Nissan Chemical Industries, Ltd. (JP) 2008-07-23 EP disclosed
US-6140338-A FOR TREATING ACUTE INFLAMMATORY DISEASES, CHRONIC INFLAMMATORY DISEASES, ACQUIRED IMMUNE DEFICIENCY SYNDROME, CANCER, ISCHEMIC REFLOW DISORDER AND/OR ARTERIOSCLEROSIS BANYU PHARMACEUTICAL, CO., LTD. (JP) 2000-10-31 US disclosed
EP-0916668-A1 CHEMOKINE RECEPTOR ANTAGONISTS BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-05-19 EP disclosed