SCHEMBL8185667

SCHEMBL8185667

O=C(/C=C/c1cnc(NCCNC(=O)c2ccc(I)cc2)c(I)c1)NOC1CCCCO1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.35
HDAC1 Q13547 2/20 0.34
IDO1 P14902 1/20 0.34
TGFBR1 P36897 1/20 0.34
GSTP1 P09211 1/20 0.33
GSTM2 P28161 1/20 0.33
PTPN1 P18031 1/20 0.32
NPC1 O15118 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
RAB9A P51151 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CCR2 P41597 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
PKM P14618 1/20 0.31
MEN1 O00255 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3223938 0.86 NPC1 (0.39) P2RX3HDAC1IDO1TGFBR1GSTP1
SCHEMBL3223927 0.86 NPC1 (0.39) P2RX3HDAC1IDO1TGFBR1GSTP1
SCHEMBL8179269 0.85 ALDH1A1 (0.34) TGFBR1SMN1; SMN2RAB9AKDM4EALDH1A1
SCHEMBL8173598 0.83 TGFBR1 (0.35) P2RX3TGFBR1
SCHEMBL8173594 0.82 TGFBR1 (0.34) TGFBR1NPC1RAB9AKDM4EALDH1A1
SCHEMBL8189381 0.81 ALDH1A1 (0.35) HDAC1TGFBR1NPC1SMN1; SMN2RAB9A
SCHEMBL8183546 0.81 KMT2A (0.37) HDAC1TGFBR1NPC1SMN1; SMN2RAB9A
SCHEMBL8185494 0.79 HDAC1 (0.45) HDAC1IDO1SMN1; SMN2HDAC6KDM4E
SCHEMBL8189383 0.78 TGFBR1 (0.34) TGFBR1SMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL8182243 0.78 MAPT (0.38) HDAC1NPC1SMN1; SMN2RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075757-A1 N-HYDROXYACRYLAMIDE COMPOUNDS ASTELLAS PHARMA INC. (JP) 2008-06-26 WO disclosed