SCHEMBL8186709

SCHEMBL8186709

c1ccc(CN2CCC(NCC3CCCCC3)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.66
BACE1 P56817 9/20 0.66
BCHE P06276 6/20 0.66
CXCR4 P61073 1/20 0.58
CXCR3 P49682 1/20 0.58
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
KDM1A O60341 1/20 0.58
MAOB P27338 1/20 0.58
DPP7 Q9UHL4 3/20 0.57
HTR2A P28223 1/20 0.56
HTR2C P28335 1/20 0.56
HTR2B P41595 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
CCR3 P51677 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3311538 0.98 ACHE (0.68) ACHEBACE1BCHECXCR4CXCR3
SCHEMBL28169202 0.89 CXCR4 (0.68) ACHEBACE1BCHECXCR4MEN1
SCHEMBL8228694 0.84 BCHE (0.57) ACHEBACE1BCHECXCR4MEN1
SCHEMBL8576045 0.84 BCHE (0.73) ACHEBACE1BCHECXCR4
SCHEMBL20183336 0.84 BCHE (0.73) ACHEBACE1BCHECXCR4
SCHEMBL31014995 0.82 BCHE (0.58) ACHEBACE1BCHEKDM1AMAOB
SCHEMBL7424698 0.81 ACHE (0.64) ACHEBACE1BCHECXCR3MEN1
SCHEMBL8805002 0.81 ACHE (0.64) ACHEBACE1BCHECXCR3MEN1
SCHEMBL9437321 0.81 ACHE (0.60) ACHEBACE1BCHECXCR4MEN1
SCHEMBL31014655 0.80 BCHE (0.61) ACHEBACE1BCHEMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156752-A Optically active 1,4-dihydropyridine compounds as bradykinin antagonists PFIZER INC (US) 2000-12-05 US disclosed
EP-0899261-A1 Optical active 1,4-dihydropyridine compounds as bradykinin antagonists PFIZER INC. (US) 1999-03-03 EP disclosed