SCHEMBL8189259

SCHEMBL8189259

CCNc1c(-c2ccccc2C)nc2c3ccccc3c(OC)cn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.42
MAPT P10636 4/20 0.40
PGK1 P00558 3/20 0.38
HSD17B10 Q99714 3/20 0.37
KDM4E B2RXH2 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CRHR1 P34998 1/20 0.36
TP53 P04637 3/20 0.36
GAA P10253 2/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CTSA P10619 1/20 0.35
USP2 O75604 1/20 0.34
CYP2D6 P10635 1/20 0.34
ALOX15 P16050 1/20 0.34
PDE2A O00408 1/20 0.34
PDE6D O43924 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8181970 0.91 CRHR1 (0.43) NR1H4MAPTHSD17B10KDM4ECYP1A2
SCHEMBL8173371 0.85 NR1H4 (0.40) NR1H4MAPTHSD17B10KDM4ECYP1A2
SCHEMBL8182713 0.82 PGK1 (0.35) NR1H4MAPTPGK1HSD17B10KDM4E
SCHEMBL8189247 0.80 NR1H4 (0.42) NR1H4MAPTHSD17B10KDM4ETP53
SCHEMBL8183161 0.79 MAPT (0.44) MAPTHSD17B10KDM4ETP53GAA
SCHEMBL8182838 0.78 NR1H4 (0.43) NR1H4MAPTCYP1A2CYP3A4GAA
SCHEMBL8173181 0.77 NR1H4 (0.41) NR1H4MAPTPGK1TP53GAA
SCHEMBL8182662 0.77 NR1H4 (0.41) NR1H4MAPTHSD17B10KDM4ETP53
SCHEMBL8172961 0.77 KMT2A (0.40) NR1H4MAPTKDM4ECYP1A2CYP3A4
SCHEMBL8187728 0.76 NR1H4 (0.40) NR1H4MAPTHSD17B10KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6103736-A SHOWING AN INHIBITORY ACTION ON GASTRIC ACID SECRETION AND A PROTECTIVE ACTION OF GASTRIC MUCOSA; 2-(HETERO)ARYL-3-AMINOIMIDAZO-(2,1-A)ISOQUINOLINES; ANTIULCER AGENTS; SHINNIPPON PHARMACEUTICAL INC. (JP) 2000-08-15 US disclosed
US-6020342-A Fused imidazo[1,2-A]pyridines SHINNIPPON PHARMACEUTICAL, INC. (JP) 2000-02-01 US disclosed
EP-0822194-A1 FUSED IMIDAZO 1,2-a]PYRIDINES Shinnippon Pharmaceutical Inc. (JP) 1998-02-04 EP disclosed