SCHEMBL8189396

SCHEMBL8189396

Cc1ccc(Oc2cccc(C=C3SC(=S)NC3=S)c2)cc1

nearest known ligand 0.78

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 9/20 0.78
MMP13 P45452 3/20 0.62
MMP3 P08254 2/20 0.62
GSK3B P49841 3/20 0.53
NAT1 P18440 2/20 0.51
AKR1B1 P15121 1/20 0.49
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8189394 1.00 ADAMTS5 (0.78) ADAMTS5MMP13MMP3GSK3BNAT1
SCHEMBL8166386 0.81 NAT1 (0.74) ADAMTS5MMP13MMP3GSK3BNAT1
SCHEMBL8166383 0.81 NAT1 (0.74) ADAMTS5MMP13MMP3GSK3BNAT1
SCHEMBL18103023 0.78 ADAMTS5 (1.00) ADAMTS5MMP13MMP3GSK3BNAT1
SCHEMBL8172889 0.78 ADAMTS5 (0.71) ADAMTS5MMP13MMP3AKR1B1TDP1
SCHEMBL8172886 0.78 ADAMTS5 (0.71) ADAMTS5MMP13MMP3AKR1B1TDP1
SCHEMBL12891792 0.78 AKR1B1 (0.81) ADAMTS5MMP13MMP3AKR1B1
SCHEMBL1247918 0.78 AKR1B1 (0.81) ADAMTS5MMP13MMP3AKR1B1
SCHEMBL1247917 0.78 AKR1B1 (0.81) ADAMTS5MMP13MMP3AKR1B1
SCHEMBL8308267 0.77 MMP13 (1.00) ADAMTS5MMP13MMP3GSK3BNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018748-A1 RHODANINE DERIVATIVES FOR THE TREATMENT AND PREVENTION OF METABOLIC BONE DISORDERS ROCHE DIAGNOSTICS GMBH (DE) 2000-04-06 WO disclosed