SCHEMBL8189587

SCHEMBL8189587

COc1ccccc1N1CCN(C2CNC2)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
DRD2 P14416 6/20 0.62
DRD3 P35462 4/20 0.62
HTR3E A5X5Y0 1/20 0.62
HTR3B O95264 1/20 0.62
ADRB1 P08588 1/20 0.62
CYP2C19 P33261 1/20 0.62
HTR3A P46098 1/20 0.62
HTR6 P50406 1/20 0.62
HTR3D Q70Z44 1/20 0.62
HTR3C Q8WXA8 1/20 0.62
SIGMAR1 Q99720 1/20 0.62
LMNA P02545 1/20 0.60
MAPT P10636 1/20 0.60
KDM4E B2RXH2 4/20 0.56
HTR1A P08908 1/20 0.55
ADRA1D P25100 1/20 0.55
ADRA1A P35348 1/20 0.55
ADRA1B P35368 1/20 0.55
HTT P42858 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3556792 0.85 DRD2 (0.68) ALDH1A1DRD2DRD3HTR3EHTR3B
SCHEMBL21204694 0.82 ALDH1A1 (0.63) ALDH1A1DRD2DRD3HTR3EHTR3B
SCHEMBL8764445 0.78 DRD2 (0.68) ALDH1A1DRD2DRD3KDM4EHTR1A
SCHEMBL3704117 0.78 KDM4E (0.63) ALDH1A1DRD2DRD3KDM4EHTR1A
SCHEMBL6635193 0.78 KDM4E (0.62) ALDH1A1DRD2DRD3MAPTKDM4E
SCHEMBL8764218 0.78 DRD2 (0.68) ALDH1A1DRD2DRD3KDM4EHTR1A
SCHEMBL8764223 0.78 DRD2 (0.68) ALDH1A1DRD2DRD3KDM4EHTR1A
SCHEMBL26418370 0.78 DRD2 (0.71) ALDH1A1DRD2DRD3HTR3EHTR3B
SCHEMBL8764013 0.77 KDM4E (0.84) ALDH1A1DRD2DRD3KDM4EHTR1A
SCHEMBL8764010 0.77 KDM4E (0.84) ALDH1A1DRD2DRD3KDM4EHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000063168-A1 SYNTHESIS OF AZETIDINE DERIVATIVES COELACANTH CHEMICAL CORPORATION (US) 2000-10-26 WO disclosed