SCHEMBL8196145

SCHEMBL8196145

COc1ccc(-c2c(C(F)F)n[nH]c2-c2ccc(SC)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40
GSK3B P49841 1/20 0.40
CDK4 P11802 4/20 0.39
CCND1 P24385 4/20 0.39
CCNE2 O96020 3/20 0.39
CCNE1 P24864 3/20 0.39
CDK2 P24941 3/20 0.39
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 3/20 0.37
MAPT P10636 2/20 0.37
GAPDH P04406 1/20 0.37
GAA P10253 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
ILK Q13418 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ALPL P05186 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640524 0.80 CCNE2 (0.38) CYP1A2GSK3BCDK4CCND1CCNE2
SCHEMBL9274671 0.80 KMT2A (0.39) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL8606259 0.80 PTGS2 (0.52) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL8926499 0.79 CCNE2 (0.35) CYP1A2GSK3BCDK4CCND1CCNE2
SCHEMBL6441245 0.75 MAPT (0.45) CYP1A1CYP1A2CYP1B1GSK3BKMT2A
SCHEMBL8195871 0.72 HTT (0.39) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL16146442 0.70 CYP1A1 (0.67) CYP1A1CYP1A2CYP1B1GSK3BKDM4E
SCHEMBL11986269 0.68 CYP1A1 (0.75) CYP1A1CYP1A2CYP1B1GSK3BKDM4E
SCHEMBL1145983 0.68 CYP1A1 (0.75) CYP1A1CYP1A2CYP1B1GSK3BKDM4E
SCHEMBL8640607 0.67 MAPK1 (0.73) KMT2AKDM4EGAAILKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed