SCHEMBL8196843

SCHEMBL8196843

Cc1cccc(C(C)C)c1NC(=O)Nc1sc2cc3c(cc2c1-c1ccccc1Cl)CCCC3

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
S1PR4 O95977 2/20 0.35
CXCL8 P10145 1/20 0.35
S1PR5 Q9H228 1/20 0.35
MAPK1 P28482 1/20 0.34
LPAR1 Q92633 1/20 0.34
PYGL P06737 1/20 0.34
NLRP3 Q96P20 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8189174 0.98 MEN1 (0.36) MEN1KMT2ACXCL8MAPK1LPAR1
SCHEMBL8198115 0.95 S1PR4 (0.39) MEN1KMT2AS1PR4S1PR5LPAR1
SCHEMBL8199588 0.93 LPAR1 (0.38) MEN1KMT2AS1PR4S1PR5LPAR1
SCHEMBL8196537 0.91 MEN1 (0.38) MEN1KMT2AMAPK1LPAR1NLRP3
SCHEMBL8197242 0.90 LPAR1 (0.38) MEN1KMT2ALPAR1NLRP3LMNA
SCHEMBL8200201 0.90 RAB9A (0.38) MEN1KMT2AS1PR4PYGLLMNA
SCHEMBL8196624 0.89 CXCL8 (0.38) MEN1KMT2AS1PR4CXCL8S1PR5
SCHEMBL8196165 0.88 LPAR1 (0.38) MEN1KMT2ALPAR1NLRP3LMNA
SCHEMBL8201678 0.86 LPAR1 (0.41) MEN1KMT2ACXCL8MAPK1LPAR1
SCHEMBL8196542 0.86 LPAR1 (0.42) MEN1KMT2AS1PR4CXCL8S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36832-E AN ANTICHOLESTEROL AGENT TREATING HYPERCHOLESTEROLEMIA NIHON NOHYAKU CO., LTD (JP) 2000-08-22 US disclosed
EP-0613894-B1 N-Heteroaryl-N'-phenylurea derivatives, their production and use NIHON NOHYAKU CO LTD (JP) 1999-05-06 EP disclosed
US-5464863-A Anticholesterol agents NIHON NOHYAKU CO., LTD. (JP) 1995-11-07 US disclosed
EP-0613894-A1 N-Heteroaryl-N'-phenylurea derivatives, their production and use NIHON NOHYAKU CO., LTD. (JP) 1994-09-07 EP disclosed