SCHEMBL8199221

SCHEMBL8199221

OC1CCN(c2cc[c]cn2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 2/20 0.39
PTPN11 Q06124 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
KCNMA1 Q12791 1/20 0.36
PDE4D Q08499 1/20 0.36
MAPT P10636 1/20 0.35
SMO Q99835 1/20 0.35
RET P07949 2/20 0.34
AURKA O14965 2/20 0.34
CDK1 P06493 2/20 0.34
CDK2 P24941 2/20 0.34
CDC7 O00311 1/20 0.34
PLK4 O00444 1/20 0.34
CHEK1 O14757 1/20 0.34
PDPK1 O15530 1/20 0.34
JAK2 O60674 1/20 0.34
ROCK2 O75116 1/20 0.34
PAK4 O96013 1/20 0.34
CHEK2 O96017 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2068713 0.90 AR (0.38) SMPD3CDK1CDK2METPDE10A
SCHEMBL2066415 0.90 AR (0.38) SMPD3CDK1CDK2METPDE10A
SCHEMBL3514940 0.90 AR (0.38) SMPD3CDK1CDK2METPDE10A
SCHEMBL4778875 0.84 HRH3 (0.37) LMNAPDE4DMAPTPDE10AKDM4E
SCHEMBL8196445 0.84 PDE10A (0.32) PDE10A
SCHEMBL8194170 0.82 MAPT (0.48) LMNAHTTMAPTLCKKDM4E
SCHEMBL8196822 0.81 PDE10A (0.41) PDE4DPDE10AMAPK8
SCHEMBL2067822 0.81 MAPT (0.36) LMNAPDE4DMAPTKDM4EALDH1A1
SCHEMBL743397 0.81 MAPT (0.40) LMNAMAPTMAPK1ALDH1A1SMN1; SMN2
SCHEMBL8199180 0.81 ALDH1A1 (0.46) PDE10AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000023444-A1 5,7-DISUBSTITUTED-4-AMINOPYRIDO[2,3-D]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2000-04-27 WO claimed
WO-2000023444-A1 5,7-DISUBSTITUTED-4-AMINOPYRIDO[2,3-D]PYRIMIDINE COMPOUNDS ABBOTT LABORATORIES (US) 2000-04-27 WO disclosed