SCHEMBL8199848

SCHEMBL8199848

Cc1ccc(CNNC(=O)OC(C)(C)C)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CCR2 P41597 5/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
P2RX7 Q99572 3/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203893 0.89 NPC1 (0.44) NPC1RAB9AALDH1A1SMN1; SMN2GAA
SCHEMBL15171404 0.85 NPC1 (0.52) NPC1RAB9ACCR2KDM4EALDH1A1
SCHEMBL7328664 0.82 HPGD (0.45) NPC1RAB9AKDM4EALDH1A1GAA
SCHEMBL6236607 0.79 GAA (0.51) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL7335575 0.77 POLB (0.46) KDM4EALDH1A1GAAMAPTPOLB
SCHEMBL13903547 0.75 GAA (0.45) NPC1RAB9AGAAL3MBTL1
SCHEMBL5015072 0.75 NPC1 (0.54) NPC1RAB9AALDH1A1SMN1; SMN2P2RX7
SCHEMBL7975698 0.75 SMN1; SMN2 (0.50) NPC1RAB9AALDH1A1SMN1; SMN2GAA
SCHEMBL6762260 0.74 MAPT (0.39) KDM4EALDH1A1SMN1; SMN2GAAMAPT
SCHEMBL18692366 0.74 APLNR (0.54) ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672678-B1 Azapeptide derivative FUJIREBIO KK (JP) 2000-10-25 EP disclosed
US-5965538-A FOR TREATING NERVOUS INFLAMMATION OF RESPIRATORY SYSTEMS, ASTHMA, BRONCHOSPASM FUJIREBIO INC. (JP) 1999-10-12 US disclosed
US-5837687-A BRONCHODILATORS, ANTIHISTAMINES AND ANTIINFLAMMATORY AGENTS; ASTHMA; ANTAGONIST OF NEUROKININ RECEPTORS FUJIREBIO INC. (JP) 1998-11-17 US disclosed
EP-0672678-A1 Azapeptide derivative FUJIREBIO Inc. (JP) 1995-09-20 EP disclosed