SCHEMBL8200409

SCHEMBL8200409

CCOC(=O)c1cc2c(C(F)(F)F)cc(OC)cc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.53
HPGD P15428 8/20 0.53
KDM4E B2RXH2 7/20 0.53
RAB9A P51151 5/20 0.53
NPC1 O15118 4/20 0.53
LMNA P02545 4/20 0.53
L3MBTL1 Q9Y468 3/20 0.53
HTT P42858 2/20 0.53
MAPT P10636 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
GAA P10253 2/20 0.46
GLA P06280 1/20 0.46
ATM Q13315 1/20 0.46
HSD17B10 Q99714 4/20 0.44
ALOX15 P16050 2/20 0.42
HRH3 Q9Y5N1 1/20 0.41
MMP13 P45452 2/20 0.41
MMP2 P08253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198168 0.92 ALDH1A1 (0.46) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL4045461 0.85 KDM4E (0.46) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL3622667 0.84 KDM4E (0.45) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL28455744 0.84 ALOX15 (0.55) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL30995200 0.83 ALDH1A1 (0.56) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL6448130 0.83 RHEB (0.52) HPGDKDM4ERHEB
SCHEMBL7879695 0.82 GABRA1 (0.48) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL703198 0.82 KDM4E (0.58) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL28844724 0.82 ALDH1A1 (0.58) ALDH1A1HPGDKDM4ERAB9ANPC1
SCHEMBL700154 0.80 KDM4E (0.51) ALDH1A1HPGDKDM4ERAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000071522-A1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS METHIONYL T-RNA SYNTHETASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 2000-11-30 WO disclosed