SCHEMBL8200539

SCHEMBL8200539

Nc1sc(Cl)cc1C(=O)NCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.55
KMT2A Q03164 2/20 0.53
NSD2 O96028 2/20 0.52
CA1 P00915 5/20 0.52
CA2 P00918 5/20 0.52
CA12 O43570 4/20 0.52
CA9 Q16790 4/20 0.52
CA3 P07451 3/20 0.52
CA6 P23280 3/20 0.52
CA5A P35218 3/20 0.52
CA7 P43166 3/20 0.52
CA13 Q8N1Q1 3/20 0.52
CA14 Q9ULX7 3/20 0.52
CA5B Q9Y2D0 3/20 0.52
CA4 P22748 2/20 0.52
TP53 P04637 3/20 0.51
MDM2 Q00987 2/20 0.51
HPGD P15428 3/20 0.50
LMNA P02545 2/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8211454 0.86 KMT2A (0.51) HSP90AA1KMT2ATP53MDM2LMNA
SCHEMBL8210407 0.83 KMT2A (0.53) KMT2ANSD2TP53HPGDLMNA
SCHEMBL20915155 0.82 GAA (0.72) KMT2ANSD2HPGDGAAMAPT
SCHEMBL8212472 0.81 ACKR3 (0.55) KMT2ATP53HPGDLMNAL3MBTL1
SCHEMBL8206773 0.81 CYP3A4 (0.53) KMT2ANSD2TP53HPGDLMNA
SCHEMBL8200561 0.80 TAAR1 (0.59) HSP90AA1KMT2ANSD2CA1CA2
SCHEMBL8206949 0.78 LMNA (0.57) KMT2AHPGDLMNAL3MBTL1APEX1
SCHEMBL8211804 0.77 LMNA (0.66) HSP90AA1KMT2ATP53HPGDLMNA
SCHEMBL8212496 0.77 GAA (0.56) KMT2AHPGDLMNAGAAAPEX1
SCHEMBL7426583 0.77 NCEH1 (0.48) TP53MDM2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed